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P1

Catalog #: 5127
1 Citation Datasheet / COA / SDS

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5127 has been discontinued.
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P1 | CAS No. 1461648-55-4 | Protein Disulphide Isomerase Inhibitors
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Description: Protein disulfide isomerase (PDI) inhibitor

Chemical Name: N-[(1,1-Dimethylethoxy)carbonyl]-L-phenylalanyl-O-(ethenylsulfonyl)-N-4-pentyn-1-yl-L-tyrosinamide

Purity: ≥98%

Product Details
Citations (1)
Reviews
Biological Activity Technical Data Background Product Datasheets Calculators

Biological Activity

P1 is a protein disulfide isomerase (PDI) inhibitor (IC50 = 1.7 μM). Inhibits proliferation of numerous cancer cell lines. Cell permeable.

Technical Data

M.Wt:
583.7
Formula:
C30H37N3O7S
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1461648-55-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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Citation for P1

The citations listed below are publications that use Tocris products. Selected citations for P1 include:

1 Citation: Showing 1 - 1

  1. Hyperglycemia exacerbates dengue virus infection by facilitating poly(A)-binding protein-mediated viral translation.
    Authors: Chia-Yi Et al.
    JCI Insight  2022;7

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