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FTI 276

Catalog #: 2406 Datasheet / COA / SDS

Discontinued Product

2406 has been discontinued.
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FTI 276 | CAS No. 1217471-51-6 | Other Transferase Inhibitors
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Description: Farnesyltransferase (FTase) inhibitor; antitumor

Chemical Name: N-[4-[2(R)-Amino-3-mercaptopropyl]amino-2-phenylbenzoyl]methionine trifluoroacetate salt

Purity: ≥95%

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Biological Activity

Ras CAAX peptidomimetic, a selective inhibitor of farnesyltransferase (FTase) that displays > 100-fold selectivity over geranylgeranyltransferase I (GGTase I) (IC50 values are 0.5 and 50 nM respectively). Blocks growth of human lung carcinoma expressing oncogenic K-Ras in nude mice.

Technical Data

M.Wt:
547.61
Formula:
C21H27N3O3S2.C2HF3O2
Solubility:
Soluble to 10 mM in water
Purity:
≥95%
Storage:
Store at -80°C
CAS No:
1217471-51-6

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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