ML 233
Chemical Name: (E)-4-Methyl-5-(((phenylsulfonyl)oxy)imino)-[1,1'-bi(cyclohexane)]-3,6-dien-2-one
Purity: ≥98%
Biological Activity
ML 233 is a non-peptide apelin receptor agonist (EC50 = 3.7 μM); exhibits >21-fold selectivity over the closely related angiotensin 1 receptor (EC50 = >79 μM).Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
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Background References
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Apelin, Elabela/Toddler, and biased agonists as novel therapeutic agents in the cardiovascular system.
Yang et al.
Trends Pharmacol Sci., 2015;36:560 -
Functional agonists of the apelin (APJ) receptor.
Khan et al.
Probe Reports from the NIH Molecular Libraries Program, 2011;
Product Datasheets
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