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VU 6015929

Catalog #: 7728 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
7728/10
7728/50
VU 6015929 | CAS No. 2442597-56-8 | DDR1/DDR2
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Description: Potent and selective discoidin domain receptor 1/2 inhibitor

Chemical Name: 4-Fluoro-3-[[[5-(1-methyl-1H-pyrazol-3-yl)-3-pyridinyl]methyl]amino]-N-[3-(trifluoromethoxy)phenyl]benzamide

Purity: ≥98%

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Biological Activity

VU 6015929 is a potent and selective discoidin domain receptor 1/2 (DDR1/2) inhibitor (IC50 = 4.67 nM and 7.39 nM for DDR1 and DDR2, respectively). VU 6015929 blocks collagen-induced DDR1 activation and collagen-IV production in HEK293 cells.

Technical Data

M.Wt:
485.43
Formula:
C24H19F4N5O2
Solubility:
Soluble to 100 mM in DMSO and to 20 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2442597-56-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets

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