WAY 207024 dihydrochloride

Name: WAY 207024 dihydrochloride
Brand: Tocris Bioscience
SKU: 3890
Price: 286 USD

Catalog #: 3890 Datasheet / COA / SDS

Discontinued Product

3890 has been discontinued.

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WAY 207024 dihydrochloride | CAS No. 872002-73-8 | GnRH Antagonist

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Description: GnRH receptor antagonist

Chemical Name: 6-[[4-[2-[4-(1,1-Dimethylethyl)phenyl]-1H-benzimidazol-7-yl]-i-piperazinyl]methyl]-quinoxaline dihydrochloride

Purity: ≥99%

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Product Details

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Biological Activity

WAY 207024 dihydrochloride is a gonadotropin releasing hormone receptor (GnRH-R) antagonist. Exhibits potent affinity (IC₅₀ values are 12 and 71 nM for human and rat GnRH receptors respectively). Lowers plasma leuteinizing hormone levels in the rat. Orally active.

Technical Data

M.Wt:

549.54

Formula:

C₃₀H₃₂N₆.2HCl

Solubility:

Soluble to 85 mM in DMSO

Purity:

≥99%

Storage:

Desiccate at RT

CAS No:

872002-73-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:

Sold for research purposes under agreement from Pfizer Inc.

Background References

Discovery of 6-({4-[2-(4-tert-butylphenyl)-1H-benzimidazol-4-yl]piperazin-1-yl}methyl)quinoxaline (WAY-207024): an orally active antagonist of the g.tropin releasing hormone receptor (GnRH-R).
Pelletier et al.
J.Med.Chem., 2009;52:214

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