BRL 52537 hydrochloride
Chemical Name: (±)-1-(3,4-Dichlorophenyl)acetyl-2-(1-pyrrolidinyl)methylpiperidine hydrochloride
Purity: ≥98%
Biological Activity
The most κ/μ-selective and among the most potent κ ligands known (25 times more potent than morphine in vivo).Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Additional Information
Background References
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High-throughput genotoxicity assay identifies antioxidants as inducers of DNA damage response and cell death.
Fox JT, Sakamuru S, Huang R
Proc. Natl. Acad. Sci. U.S.A., 2012;109(14):5423-8. -
(2S)-1-(Arylacetyl)-2-(aminomethyl)piperidine derivatives: novel, highly selective κ opioid analgesics.
Vecchietti et al.
J.Med.Chem., 1991;34:397
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Citation for BRL 52537 hydrochloride
The citations listed below are publications that use Tocris products. Selected citations for BRL 52537 hydrochloride include:
1 Citation: Showing 1 - 1
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Label-free integrative pharmacology on-target of opioid ligands at the opioid receptor family.
Authors: Morse Et al.
BMC Pharmacol Toxicol 2013;14:17
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