Tianeptine sodium salt

Tocris Bioscience | Catalog # 1972

Selective facilitator of 5-HT uptake; antidepressant
Tocris Bioscience
Discontinued Product
1972 has been discontinued. View all 5-HT Transporter Compounds products.

Key Product Details

Description

Selective facilitator of 5-HT uptake; antidepressant
View all 5-HT Transporter Compounds »

Product Description

Tianeptine sodium salt is a selective facilitator of 5-HT uptake in vitro and in vivo. Has no affinity for a wide range of receptors, including 5-HT and dopamine (IC50 > 10 μM) and has no effect on noradrenalin or dopamine uptake. Antidepressant, analgesic and neuroprotective following systemic administration in vivo.

Product Specifications for Tianeptine sodium salt

Molecular Weight

458.93

Formula

C21H24ClN2NaO4S

Storage

Desiccate at RT

Purity

≥99% (HPLC)

Chemical Name

7-[(3-Chloro-6,11-dihydro-6-methyl-5,5-dioxidodibenzo[c,f][1,2]thiazepin-11-yl)amino]heptanoic acid sodium salt

CAS Number

30123-17-2

PubChem ID

23663953

InChI Key

ZLBSUOGMZDXYKE-UHFFFAOYSA-M

SMILES

[Na+].CN1C2=CC=CC=C2C(NCCCCCCC([O-])=O)C2=CC=C(Cl)C=C2S1(=O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Solubility

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 45.89 100
DMSO 4.58 10

Preparing Stock Solutions for Tianeptine sodium salt

The following data is based on the product molecular weight 458.93.

Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which all affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 2.18 mL 10.89 mL 21.79 mL
5 mM 0.44 mL 2.18 mL 4.36 mL
10 mM 0.22 mL 1.09 mL 2.18 mL
50 mM 0.04 mL 0.22 mL 0.44 mL

Calculators

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Background References

References are publications that support the biological activity of the product. See our Citations tab to view 115 publications citing the usage of this product.

Product Documents for Tianeptine sodium salt

Certificate of Analysis

To download a Certificate of Analysis, please enter a lot or batch number in the search box below.

Product Specific Notices for Tianeptine sodium salt

For research use only

Citations for Tianeptine sodium salt

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