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BMS 466442

Catalog #: 6878 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
6878/10
BMS 466442 | CAS No. 1598424-76-0 | Other Ion Pump/Transporter Inhibitors
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Description: Potent and selective inhibitor of asc-1

Chemical Name: N-[[5-Methoxy-6-(phenylmethoxy)-1H-indol-2-yl]carbonyl]-1-(phenylmethyl)-L-histidine methyl ester

Purity: ≥98%

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Biological Activity

BMS 466442 is a potent and selective asc-1 (alanine-serine-cysteine-1) transporter inhibitor (IC50 values are 20 and 37 nM in rat primary cortical cultures and HEK cells expressing asc-1 respectively). Displays >1000-fold selectivity for asc-1 over LAT-2 and ASCT-2. This compound is unsuitable for in vivo studies.

Technical Data

M.Wt:
538.6
Formula:
C31H30N4O5
Solubility:
Soluble to 100 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
1598424-76-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

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