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(±)-CP 47497

Catalog #: 3500 Datasheet / COA / SDS

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3500 has been discontinued.
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(±)-CP 47497 | CAS No. 70434-82-1 | Cannabinoid R1/CB1 Agonists
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Description: Potent CB1 agonist

Chemical Name: rel-5-(1,1-Dimethylheptyl)-2-[(1R,3S)-3-hydroxycyclohexyl]phenol

Purity: ≥98%

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Biological Activity

Potent CB1 receptor agonist (Ki = 2.2 nM). Exhibits analgesic, motor depressant, anticonvulsant and hypothermic effects in vivo.

Technical Data

M.Wt:
318.49
Formula:
C21H34O2
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in ethanol
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
70434-82-1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

  1. Cannabimimetic activity from CP-47,497, a derivative of 3-phenylcyclohexanol.
    Weissman et al.
    J.Pharmacol.Exp.Ther., 1982;223:516
  2. Structure-activity relationships for cannabinoid receptor-binding and analgesic activity: studies of bicyclic cannabinoid analogs.
    Melvin et al.
    Mol.Pharmacol., 1993;44:1008
  3. Synthesis and pharmacology of 1-deoxy analogs of CP-47,497 and CP-55,940.
    Huffman et al.
    Bioorg.Med.Chem., 2008;16:322
  4. Direct On-Chip Differentiation of Intestinal Tubules from Induced Pluripotent Stem Cells
    E Naumovska, G Aalderink, C Wong Valen, K Kosim, A Nicolas, S Brown, P Vulto, KS Erdmann, D Kurek
    Int J Mol Sci, 2020;21(14):.

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