Droperidol
Discontinued Product
Chemical Name: 1-[1-[4-(4-Fluorophenyl)-4-oxobutyl]-1,2,3,6-tetrahydro-4-pyridinyl]-1,3-dihydro-2H-benzimidazol-2-one
Purity: ≥98%
Biological Activity
Droperidol is a D2 receptor antagonist. Also exhibits affinity for 5-HT, α-adrenergic and histamine receptors,and hERG channels. Antipsychotic and antiemetic.Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
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Relationship of neuroleptic drug effects at brain DA, serotonin, alpha-adrenergic, and histamine receptors to clinical potency.
Peroutka and Synder
Am.J.Psychiatry, 1980;137:1518 -
A two-state homology model of the hERG K+ channel: application to ligand binding.
Rajamani et al.
Bioorg.Med.Chem.Lett., 2005;15:1737
Product Datasheets
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