LY 2087101
Chemical Name: [2-[(4-Fluorophenyl)amino]-4-methyl-5-thiazolyl]-3-thienylmethanone
Purity: ≥98%
Biological Activity
LY 2087101 is an allosteric potentiator of α7, α4β2 and α4β4 nAChRs; displays selectivity against α3β4 nAChRs. Thought to potentiate agonist-evoked α7 responses by binding within the nAChR transmembrane region.Technical Data
The technical data provided above is for guidance only.
For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Background References
-
Identification and pharmacological profile of a new class of selective nicotinic acetylcholine receptor potentiators.
Broad et al.
J.Pharmacol.Exp.Ther., 2006;318:1108
Product Datasheets
Reconstitution Calculator
Molarity Calculator
Citation for LY 2087101
The citations listed below are publications that use Tocris products. Selected citations for LY 2087101 include:
1 Citation: Showing 1 - 1
-
Studying Nicotinic Acetylcholine Receptors Using the IonFlux™ Microfluidic-Based Automated Patch-Clamp System with Continuous Perfusion and Fast Solution Exchange.
Authors: Haiyang Et al.
Curr Protoc Pharmacol 2020;88:e73
FAQs
No product specific FAQs exist for this product, however you may
View all Small Molecule FAQsReviews for LY 2087101
There are currently no reviews for this product. Be the first to review LY 2087101 and earn rewards!
Have you used LY 2087101?
Submit a review and receive an Amazon gift card.
$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image
$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image
