SR 16584

Catalog #: 4424 Datasheet / COA / SDS

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SR 16584 | CAS No. 1150153-86-8 | Additional Nicotinic Receptor Antagonists

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Description: Selective α3β4 nAChR antagonist

Chemical Name: 1,3-Dihydro-1-(3-exo)-9-methyl-9-azabicyclo[3.3.1]non-3-yl]-2H-indol-2-one

Purity: ≥98%

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Biological Activity

SR 16584 is a selective α3β4 nAChR antagonist (IC₅₀ = 10.2 μM). Selectively binds α3β4 over α4β2 and α7 subtypes (K_i values are 0.508, >100 and >100 μM, respectively).

Technical Data

M.Wt:

270.37

Formula:

C₁₇H₂₂N₂O

Solubility:

Soluble to 100 mM in DMSO

Purity:

≥98%

Storage:

Store at -20°C

CAS No:

1150153-86-8

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Background References

Novel α3β4 nicotinic acetylcholine receptor-selective ligands. Discovery, structure-activity studies, and pharmacological evaluation.
Zaveri et al.
J.Med.Chem., 2012;53:8187

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