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TP 238

Catalog #: 6670 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
6670/10
TP 238 | CAS No. 2415263-05-5 | Bromodomain Inhibitors
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Description: CECR2 and BPTF/FALZ inhibitor

Chemical Name: N-[(3-(1H)-Pyrazol-1-yl)propyl)-6-(4-(3-(dimethylamino)propoxy)phenyl)-2-(methylsulfonyl)pyrimidin-4-amine hydrochloride

Purity: ≥98%

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Biological Activity

TP 238 is a cat eye syndrome chromosome region, candidate 2 (CECR2) and bromodomain PHD finger transcription factor (BPTF/FALZ) inhibitor (IC50 values are 10-30 and 100-350 nM, respectively).

A concentration of no more than 2 μM is recommended for use in cellular assays.

Technical Data

M.Wt:
495.04
Formula:
C22H30N6O<sub>3S.HCl
Solubility:
Soluble to 100 mM in DMSO and to 100 mM in water
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2415263-05-5

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the TP 238 probe summary on the SGC website.

Product Datasheets

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