Home / mAChR M5 Antagonists / VU 6019650

VU 6019650

Catalog #: 8055 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
8055/50
8055/10
VU 6019650 | CAS No. 2926782-31-0 | mAChR M5 Antagonists
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Description: M5 receptor antagonist

Chemical Name: (3R,4S)-rel-1-[(2,3-Dihydro-5-benzofuranyl)sulfonyl]-3-fluoro-4-[[(1-methyl-1H-imidazol-2-yl)thio]methyl]piperidine

Purity: ≥98%

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Biological Activity

VU 6019650 is a potent and selective M5 receptor antagonist (hM5 IC50 = 36 nM). Exhibits >100-fold selectivity over human and rat M1-4. In vivo, VU 6019650 inhibits the reward effects of oxycodone and reduces oxycodone self-administration in rats. VU 6019650 is blood brain barrier penetrant.

Technical Data

M.Wt:
411.51
Formula:
C18H22FN3O3S2
Solubility:
Soluble to 50 mM in DMSO
Purity:
≥98%
Storage:
Store at -20°C
CAS No:
2926782-31-0

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license from Vanderbilt University

Product Datasheets

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