Home / Histone Demethylase Inhibitors / GSK J2

GSK J2

Catalog #: 4688 Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
4688/10
4688/50
GSK J2 | CAS No. 1394854-52-4 | Histone Demethylase Inhibitors
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Description: Inactive isomer of GSK J1 (Cat. No. 4593)

Chemical Name: N-[2-(3-Pyridinyl)-6-(1,2,4,5-tetrahydro-3H-3-benzazepin-3-yl)-4-pyrimidinyl]-β-alanine ethyl ester

Purity: ≥98%

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Biological Activity

GSK J2 is an inactive control of GSK J1 (IC50 > 100 μM for inhibition of JMJD3/UTX).

Cell permeable ester derivative, GSK J5 and Active Analog also available.

Technical Data

M.Wt:
389.45
Formula:
C22H23N5O2
Solubility:
Soluble to 100 mM in DMSO and to 50 mM in 1eq. HCl
Purity:
≥98%
Storage:
Desiccate at RT
CAS No:
1394854-52-4

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
This compound is supplied in conjunction with the Structural Genomics Consortium. For further details of GSK J2, an inactive isomer of GSK J1, please visit the GSK J1 probe summary on the SGC website.
Other Product-Specific Information:

Product Datasheets

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