Home / KISS-Derived Peptide Receptor Antagonists / Kisspeptin 234

Kisspeptin 234

Catalog #: 3881
4 Citations Datasheet / COA / SDS
Catalog # Availability Size / Price Qty
3881/1
Kisspeptin 234
1 Image
Description: Kisspeptin receptor antagonist; kisspeptin 10 (Cat. No. 2570) analog

Purity: ≥95%

Product Details
Citations (4)
Supplemental Products
Reviews
Biological Activity Technical Data Additional Information Background Product Datasheets Calculators

Biological Activity

Kisspeptin 234 is a kisspeptin receptor (KISS1, GPR54) antagonist; kisspeptin-10 (Cat. No. 2570) analog. Inhibits kisspeptin-10 stimulation of inositol phosphate (IP) (IC50 = 7 nM) and release of gonadotrophin-releasing hormone (GnRH).

Technical Data

M.Wt:
1295.42
Formula:
C63H78N18O13
Sequence:
Ac-ANWNGFGWRF-NH2

(Modifications: Ala-1 = D-Ala & N-terminal Ac, Trp-8 = D-Trp, Phe-10 = C-terminal amide)

Solubility:
Soluble to 1 mg/ml in water
Purity:
≥95%
Storage:
Store at -20°C
CAS No:
1145998-81-7

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.

Additional Information

Licensing Caveats:
Sold under license

Product Datasheets

COA view current batch
Or select another batch:
View Batch
SDS
Reconstitution Calculator
Molarity Calculator

Reconstitution Calculator

The reconstitution calculator allows you to quickly calculate the volume of a reagent to reconstitute your vial. Simply enter the mass of reagent and the target concentration and the calculator will determine the rest.

=
÷

Molarity Calculator

=
x
x
g/mol

*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and CoA (available online).

Citations for Kisspeptin 234

The citations listed below are publications that use Tocris products. Selected citations for Kisspeptin 234 include:

4 Citations: Showing 1 - 4

  1. Kisspeptins inhibit human airway smooth muscle proliferation.
    Authors: Y S Et al.
    JCI Insight  2022;7
  2. Kisspeptin-54 attenuates oxidative stress and neuronal apoptosis in early brain injury after subarachnoid hemorrhage in rats via GPR54/ARRB2/AKT/GSK3β signaling pathway.
    Authors: Lei Et al.
    Free Radic Biol Med  2021;171:99-111
  3. The pregnant mouse uterus exhibits a functional kisspeptin/KISS1R signaling system on the day of embryo implantation.
    Authors: Fayazi Et al.
    Am J Physiol Renal Physiol  2015;13:105
  4. GPR54-dependent stimulation of luteinizing hormone secretion by neurokinin B in prepubertal rats.
    Authors: Grachev Et al.
    Reprod Biol Endocrinol  2012;7:e44344

FAQs

No product specific FAQs exist for this product, however you may

View all Peptide FAQs

Reviews for Kisspeptin 234

There are currently no reviews for this product. Be the first to review Kisspeptin 234 and earn rewards!

Have you used Kisspeptin 234?

Submit a review and receive an Amazon gift card.

$25/€18/£15/$25CAN/¥75 Yuan/¥2500 Yen for a review with an image

$10/€7/£6/$10 CAD/¥70 Yuan/¥1110 Yen for a review without an image

Submit a Review
Tocris Bioscience is the leading supplier of novel and exclusive tools for life science research with over 30 years' experience in the industry. Tocris is a Bio-Techne brand.